Calbiochem™ Haspin Kinase Inhibitor, Chr-6494, Each

Details:

A cell-permeable indazolylimidazopyridazinamine compound that acts as a potent and reversible inhibitor of histone kinase haspin activity (ic50 = 2nm) with moderate selectivity over trka, gsk-3β, pim1, cdk1/b and cdk2/a (% inhibition at 100nm = 58, 48, 36, 34 and 33, respectively) among a panel of 27-kina