518-831-8000 sales@utechproducts.com

Bms 195614, Selective Rarα Antagonist, Each

528.53

Details:

BMS 195614 is a neutral retinoic acid receptor (RAR) α-selective antagonist (Ki = 2.5 nM). Displays no significant effect on nuclear receptor corepressor (NCoR) binding; moderately decreases SMRT binding to RAR. Antagonizes agonist-induced coactivator (CoA) recruitment.

Additional Information

SKU 1614637
UOM Each
UNSPSC 41116105
Manufacturer Part Number 3660/10