Sarpogrelate Hydrochloride, Selective 5-Ht2a Antagonist, Each

Details

Sarpogrelate hydrochloride is a selective 5-ht2a receptor antagonist (pki values are 8.52, 7.43 And 6.57 For 5-ht2a, 5-ht2c and 5-ht2b receptors respectively). Displays selectivity over 5-ht1, 5-ht3, 5-ht4 h1, h2, m3, α1-adrenergic, α2-adrenergic and β-adrenergic receptors. Displays cardioprotective activity in vivo.